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5-Amino-1MQ is commonly studied in the context of NNMT inhibition, NAD+ salvage pathway modulation, adipocyte biology, and metabolic flux in preclinical models
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Oncology work is a separate, unrelated thread NNMT is also overexpressed in a number of tumours, and 5-amino-1-methylquinolinium has been used as a tool compound in cancer biology — showing concentration- and time-dependent antiproliferative activity against HeLa cervical cancer cells in vitro [10] , and reducing tumour growth while enhancing the apoptotic effect of an anti-PD-L1 antibody in bladder cancer mouse models [11]
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